Friday, June 3, 2011

Epsilon-aminocaproic acid vs Antidiuretic Hormone

Methadone works weaker, but the duration of morphine given by mouth. Eliminate respiratory depression, eyforiziruyuschee effect and other effects of opioid analgesics. Apply trimeperidin myocardial infarction, malignant tumors, trauma, as well as pain associated with spasm of smooth muscles of internal organs. Little effect on respiration. Methadone is used to order replacement therapy in Negative treatment of drug dependence to opioids. a2Adrenomimetik clonidine (clonidine), reduces pain, apparently due to stimulation adrenoretseptor and enhance descending inhibitory influences on the conduct pain impulses Nasotracheal Tube the putting afferent paths brain. Trimeperidin contraindicated in respiratory depression. Heroin is rapidly hydrolyzed in the body into an active 6monoatsetilmorfin, which is the same as heroin, vysokolipofilen, easily penetrates Dead on Arrival central nervous system and is transformed into morphine. Stimulate oretseptor (sigmaretseptor), and therefore the their application can be dysphoria, hallucinations, tachycardia, increased blood pressure. In contrast, morphine omnopon does not cause spasm of smooth muscles, as it contains alkaloids of isoquinoline series - papaverine and nartsein having myotropic inflammatory properties. Fentanyl is stronger than morphine, depresses the respiratory center. Stimulates the reduction of the myometrium. Fentanyl Amino Acids talamonal can be applied to eliminating putting pain of injuries. Tolerance and physical dependence to methadone develops more slowly, after withdrawal of methadone withdrawal is expressed to a lesser extent, but lasting than in comparison with morphine. Analgesic effects, sufficient to for short surgical procedures, providing ketamine (ketalar), which blocks the receptors of excitatory amino acids (NMDApetseptor). Tramadol (Tramal) has the properties putting opioid analgesics (stimulates myuretseptor), and furthermore, breaks back neuronal capture of norepinephrine and serotonin, ie, activates noradrenergic and serotonergic transmission, and may enhance downstream inhibitory effects on the conduct pain impulses. On chemical structure and properties similar to sufentanil with fentanyl, which exceed fentanyl on activity. On analgesic effect of morphine is inferior. Due to the high content of morphine omnopon applied for the same indications as morphine. Length of fentanyl 20-30 min. The drug is administered intravenously or intramuscularly. Plaster stick to a healthy area of skin at 72 h. However, the pharmacological properties of these drugs are similar to morphine. The highest daily dose of paracetamol - 4 in putting of overdose paracetamol is the possibility of severe liver damage (necrosis) because of the toxic metabolite of paracetamol - Natsetilpbenzohinonimina (at therapeutic doses of paracetamol, this metabolite is rapidly inactivated by glutathione). Morphine content is omnopone 48-50%. As a result, when using heroin euphoria develops faster and more pronounced than with morphine. Codeine may be effective in acute infectious diarrhea. Used fentanyl for sedation before surgery, for pain in the postoperative period. In most countries, the use of this drug is prohibited. To accelerate the elimination of morphine from organism used forced diuresis or peritoneal dialysis. To eliminate chronic pain use transdermal therapeutic system (patch) with fentanyl. In case of deep respiratory depression have resorted to artificial ventilation. Naltrexone acts in 2448 h, he was appointed interior in the treatment of drug addicts to prevent eyforiziruyuschego action of morphine, heroin and other opioids. On the chemical structure of morphine differ trimeperidin and fentanyl - Derivatives phenylpiperidine. When the pain associated with spasm of smooth muscles, such as kidney and liver colic, omnopon has an advantage over Benign Prostatic Hyperplasia On pharmacological properties similar to morphine, heroin (diacetylmorphine) and codeine (metilmorfin). Opioid antagonists analgesics - naloxone and naltrexone block mainly tsretseptor and to a lesser extent kretseptor and 8retseptor. At the same time, codeine is more suitable for use inside (Bioavailability of codeine 50%).
 

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